Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12554 | PROTAC EED degrader-2 | Others | Others |
PROTAC EED degrader-2 is a PROTAC targeting EED (pKD of 9.27),is a inhibitor of polycomb repressive complex 2 (PRC2) with pIC50 of 8.11. | |||
T13954 |
UNC6852
|
Histone Methyltransferase; Ligands for Target Protein for PROTAC | Chromatin/Epigenetic; PROTAC |
UNC6852 包含一个 EED 配体 (IC50 = 247 nM) 和一个 von Hippel-Lindau 配体,是一种基于 PROTAC 的特异性多梳抑制复合物 2 (PRC2) 降解剂。 | |||
T13765 |
MAK683-CH2CH2COOH
|
Others | Others |
MAK683-CH2CH2COOH 与 EED (胚胎外胚层发育蛋白) 结合。基于MAK683-CH2CH2COOH 和 E3 泛素连接酶的 VHL 配体,设计了靶向EED 的PROTACs, PROTAC EED degrader-1 和 PROTAC EED degrader-2 。 | |||
T73945 | MAK683-CH2CH2COOH hydrochloride | ||
MAK683-CH2CH2COOH 与 EED (胚胎外胚层发育蛋白) 结合。MAK683-CH2CH2COOH 和 E3 泛素连接酶的 VHL 配体设计了 PROTACEED degrader-1 和 PROTACEED degrader-2 。 | |||
T12553 |
PROTAC EED degrader-1
|
Others | Others |
PROTAC EED degrader-1 is a PROTAC targeting EED (pKD = 9.02), is a inhibitor of polycomb repressive complex 2 (PRC2) with pIC50 of 8.17. |